A fluorine scan of non-peptidic inhibitors of neprilysin: Fluorophobic and fluorophilic regions in an enzyme active site
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Author / Producer
Date
2008
Publication Type
Journal Article
ETH Bibliography
yes
Citations
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Rights / License
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Publication status
published
Editor
Book title
Journal / series
Volume
129 (9)
Pages / Article No.
852 - 865
Publisher
Elsevier
Event
Edition / version
Methods
Software
Geographic location
Date collected
Date created
Subject
Neprilysin; Fluorine interactions; Medicinal chemistry; pKa value; Benzimidazole
Organisational unit
03344 - Diederich, François (emeritus)
Notes
Received 26 January 2008, Revised 19 February 2008, Accepted 19 February 2008, Available online 23 February 2008.