Leveraging the Pre-DFG Residue Thr-406 To Obtain High Kinase Selectivity in an Aminopyrazole-Type PAK1 Inhibitor Series


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Date

2015

Publication Type

Journal Article

ETH Bibliography

yes

Citations

Altmetric
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Data

Rights / License

Publication status

published

Editor

Book title

Volume

6 (6)

Pages / Article No.

711 - 715

Publisher

American Chemical Society

Event

Edition / version

Methods

Software

Geographic location

Date collected

Date created

Subject

Pre-DFG residue; PAK1 kinase; Aminopyrazole

Organisational unit

03344 - Diederich, François (emeritus) check_circle

Notes

Received 11 April 2015, Accepted 20 May 2015, Published online 20 May 2015.

Funding

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