The Substrate-Activity-Screening methodology applied to receptor tyrosine kinases
A proof-of-concept study
dc.contributor.author
Chapelat, Julien
dc.contributor.author
Berst, Frédéric
dc.contributor.author
Marzinzik, Andreas L.
dc.contributor.author
Moebitz, Henrik
dc.contributor.author
Drueckes, Peter
dc.contributor.author
Trappe, Joerg
dc.contributor.author
Fabbro, Doriano
dc.contributor.author
Seebach, Dieter
dc.date.accessioned
2017-06-10T13:04:03Z
dc.date.available
2017-06-10T13:04:03Z
dc.date.issued
2012-11
dc.identifier.issn
0223-5234
dc.identifier.issn
1768-3254
dc.identifier.other
10.1016/j.ejmech.2012.08.038
dc.identifier.uri
http://hdl.handle.net/20.500.11850/62277
dc.language.iso
en
dc.publisher
Elsevier
dc.subject
Kinase inhibitor
dc.subject
Substrate-Activity-Screening
dc.subject
Proteineprotein interactions
dc.subject
MichaeliseMenten kinetics
dc.subject
Insulin-like Growth Factor 1 Receptor
dc.title
The Substrate-Activity-Screening methodology applied to receptor tyrosine kinases
dc.type
Journal Article
ethz.title.subtitle
A proof-of-concept study
ethz.journal.title
European Journal of Medicinal Chemistry
ethz.journal.volume
57
ethz.journal.abbreviated
EJMCA
ethz.pages.start
1
ethz.pages.end
9
ethz.notes
Received 2 May 2012, Accepted 26 August 2012, Available online 4 September 2012.
ethz.identifier.nebis
001485318
ethz.publication.place
Paris
ethz.publication.status
published
ethz.leitzahl
ETH Zürich::00002 - ETH Zürich::00012 - Lehre und Forschung::00007 - Departemente::02020 - Dep. Chemie und Angewandte Biowiss. / Dep. of Chemistry and Applied Biosc.::02514 - Laboratorium für Organische Chemie / Laboratory of Organic Chemistry::03492 - Hilvert, Donald (emeritus) / Hilvert, Donald (emeritus)
ethz.leitzahl.certified
ETH Zürich::00002 - ETH Zürich::00012 - Lehre und Forschung::00007 - Departemente::02020 - Dep. Chemie und Angewandte Biowiss. / Dep. of Chemistry and Applied Biosc.::02514 - Laboratorium für Organische Chemie / Laboratory of Organic Chemistry::03492 - Hilvert, Donald (emeritus) / Hilvert, Donald (emeritus)
ethz.date.deposited
2017-06-10T13:05:12Z
ethz.source
ECIT
ethz.identifier.importid
imp593650423851b85177
ethz.ecitpid
pub:98951
ethz.eth
yes
ethz.availability
Metadata only
ethz.rosetta.installDate
2017-07-12T21:34:11Z
ethz.rosetta.lastUpdated
2021-02-14T09:57:40Z
ethz.rosetta.versionExported
true
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Journal Article [128876]